Eplerenone
Eplerenone

2.55
A generic alternative indicated for Heart and Blood Pressure. This formulation supports the blockade of hormone receptors that contribute to fluid retention and elevated pressure.


Ingredient
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Eplerenone
Reference Brand
Inspra
Product Origin
Generic Product
Reference Manufacturer
Pfizer
Product Form
Tablet
Regulatory Classification
Rx
Primary Category
Heart Health
Product Category
Aldosterone Antagonist
Pharmacological Class
Selective Aldosterone Receptor Antagonist
Manufacturer Description
Formulated to manage heart failure and address hypertension by regulating mineral balance to alleviate cardiac strain and support improved cardiovascular survival outcomes.
Mechanism of Action
Eplerenone blocks the effects of aldosterone, a hormone that causes the body to retain salt and water. By preventing this, it helps the heart pump more easily and lowers blood pressure while reducing heart tissue scarring.
Route of Administration
Oral
Onset Time
Steady state in 2 days
Duration
24 hours
Contraindications
High blood potassium levels, Severe kidney impairment, Strong CYP3A inhibitors, Diabetes with microalbuminuria
Severe Adverse Events
Severe hyperkalemia, Kidney failure, Severe allergic reactions, Heart rhythm changes, Chest pain
Common Side Effects
Dizziness, Fatigue
Uncommon Side Effects
Headache, Diarrhea, Nausea, Increased potassium, Cough, Flu-like symptoms
Drug Interactions
Ketoconazole, Itraconazole, Ritonavir, Potassium supplements, ACE inhibitors, NSAIDs
Pregnancy Safety Warnings
Use only if benefit justifies potential risk to the fetus.
Age Restrictions
Safety not established in children.
Storage Guidelines
Store at room temperature.
Related Products
Information for Eplerenone is sourced from established medical standards and updated frequently. It is provided for general reference and should be confirmed with a healthcare professional before use.
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