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Isentress
Isentress

7.29
A generic alternative indicated for HIV. Therapy facilitates the inhibition of viral integrase to support stable immune system function.
Ingredient
Raltegravir Potassium
Category
HIV
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Raltegravir Potassium
Reference Brand
Raltegravir
Product Origin
Generic Alternative
Reference Manufacturer
Merck Sharp & Dohme
Product Form
Tablet, Chewable Tablet, Granules
Regulatory Classification
Rx
Primary Category
Infection Treatment
Product Category
Antiviral (Integrase Inhibitor)
Pharmacological Class
Integrase Inhibitor
Manufacturer Description
Indicated to alleviate HIV-1 infection severity by addressing viral integration to support immune health and mitigate the risk of clinical disease progression effectively.
Mechanism of Action
Raltegravir inhibits the HIV integrase enzyme. HIV needs this enzyme to insert its genetic code into the DNA of the host's cells. By blocking this step, the virus is unable to replicate or infect new immune cells.
Route of Administration
Oral
Onset Time
Steady state in 2 days
Duration
12–24 hours (formulation dependent)
Contraindications
Hypersensitivity to raltegravir
Severe Adverse Events
Severe skin reactions (SJS), Muscle breakdown (Rhabdomyolysis), Liver failure, Severe psychiatric symptoms (Depression), Immune reconstitution syndrome
Common Side Effects
Headache, Nausea
Uncommon Side Effects
Insomnia, Fatigue, Dizziness, Diarrhea, Muscle pain
Drug Interactions
Rifampin, Phenytoin, Antacids, Calcium supplements, Warfarin
Pregnancy Safety Warnings
Generally considered safe for use during pregnancy; preferred integrase inhibitor in many guidelines.
Age Restrictions
Approved for infants weighing at least 2 kg.
Storage Guidelines
Store at room temperature in the original container.
Related Products
Dolutegravir, Elvitegravir, Bictegravir
Information for Isentress is sourced from established medical standards and updated frequently. It is provided for general reference and should be confirmed with a healthcare professional before use.
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