Tolvaptan
Tolvaptan

5.02
A clinical formulation indicated for Hormone Therapy. This medicine supports the balance of electrolytes and fluid levels by managing vasopressin activity in the body.


Ingredient
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Tolvaptan
Reference Brand
Samsca
Product Origin
Generic Product
Reference Manufacturer
Otsuka Pharmaceutical
Product Form
Tablet
Regulatory Classification
Rx
Primary Category
Hormone Therapy, Heart Health
Product Category
Aquaretic
Pharmacological Class
Vasopressin V2 Receptor Antagonist
Manufacturer Description
Intended to manage fluid overload by addressing electrolyte imbalances to alleviate low blood sodium and support kidney health in polycystic disease patients effectively.
Mechanism of Action
Tolvaptan blocks the action of vasopressin in the kidneys. This prevents the body from retaining too much water, allowing the kidneys to excrete excess fluid without losing essential electrolytes like sodium.
Route of Administration
Oral
Onset Time
2–4 hours
Duration
24 hours
Contraindications
Need to increase sodium rapidly, Inability to sense thirst, Anuria, Severe liver disease, Strong CYP3A inhibitors
Severe Adverse Events
Severe liver injury, Osmotic demyelination syndrome, Dehydration, Gastrointestinal bleeding, Severe allergic reactions
Common Side Effects
Thirst, Dry mouth
Uncommon Side Effects
Frequent urination, Constipation, Nausea, Dizziness
Drug Interactions
Ketoconazole, Clarithromycin, Ritonavir, Rifampin, Digoxin
Pregnancy Safety Warnings
Use only if benefit justifies potential risk to the fetus.
Age Restrictions
Not for use in children.
Storage Guidelines
Store at room temperature in the original pack.
Related Products
Conivaptan, Furosemide
Information for Tolvaptan is sourced from established medical standards and updated frequently. It is provided for general reference and should be confirmed with a healthcare professional before use.
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